Asivatrep (PAC-14028)

Name: Asivatrep (PAC-14028); MyBioSource
Brand: MyBioSource
SKU: MBS3600042
Price: 425 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3600042

Asivatrep (PAC-14028) is a potent, selective TRPV1 antagonist with IC50 of 55 nM against capsaicin-induced Ca2+ influx in rat DRG neurons. More details

$425 / 5 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Asivatrep, Biochemical

Full Product Name

Asivatrep

Product Synonym Names

PAC-14028; PAC14028

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

491.4747

Suitability

DMSO: >=28mg/mL

Target

TRP/TRPV Channel

Receptor

TRP/TRPV Channel

Chemical Name

2-Propenamide, N-[(1R)-1-[3, 5-difluoro-4-[(methylsulfonyl)amino]phenyl]ethyl]-3-[2-propyl-6-(trifluoromethyl)-3-pyridinyl]-, (2E)

SMILES

O=C(N[C@@H](C1=CC(F)=C(NS(=O)(C)=O)C(F)=C1)C)/C=C/C2=CC=C(C(F)(F)F)N=C2CCC

Molecular Formula

C21H22F5N3O3S

CAS Number

1005168-10-4

Product Categories/Family for Asivatrep biochemical

Dermatitis; Membrane Transporter/Ion Channel; Inflammation/Immunology

Product References and Citations for Asivatrep biochemical

1. Yun JW, et al. J Dermatol Sci. 2011 Apr; 62 (1):8-15.
2. Yun JW, et al. J Invest Dermatol. 2011 Jul; 131 (7):1576-9.
3. Lim KM, et al. Arch Pharm Res. 2012 Mar; 35 (3):393-6.

Other Notes

Small volumes of Asivatrep biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Asivatrep purchase

MBS3600042 is a biochemical targeting Asivatrep.