GSK-2140944 (Gepotidacin)

Name: GSK-2140944 (Gepotidacin); MyBioSource
Brand: MyBioSource
SKU: MBS3600308
Price: 320 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3600308

GSK-2140944 (Gepotidacin) is a novel potent, selective bacterial type II topoisomerase inhibitor in development for the treatment of conventional and biothreat pathogens. More details

$320 / 2 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

GSK-2140944, Biochemical

Full Product Name

GSK-2140944

Product Synonym Names

Gepotidacin; GSK2140944

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

448.527

Suitability

DMSO: 7.14mg/mL (15.92mM)

Target

Antibacterial

Receptor

Antibacterial

Chemical Name

(2R)-2-[[4-[[(3, 4-Dihydro-2H-pyrano[2, 3-c]pyridin-6-yl)methyl]amino]-1-piperidinyl]methyl]-1, 2-dihydro-3H, 8H-2a, 5, 8a-triazaacenaphthylene-3, 8-dione

SMILES

O=C(C=NC(C=C1)=C23)N3[C@H](CN4CCC(NCC(N=C5)=CC6=C5OCCC6)CC4)CN2C1=O

Molecular Formula

C24H28N6O3

CAS Number

1075236-89-3

Product Categories/Family for GSK-2140944 biochemical

Bacterial Infection; GPCR/G Protein; Infection

Product References and Citations for GSK-2140944 biochemical

1. Bax BD, et al. Nature. 2010 Aug 19; 466 (7309):935-40.
2. Biedenbach DJ, et al. Antimicrob Agents Chemother. 2016 Jan 4; 60 (3):1918-23.
3. So W, et al. Antimicrob Agents Chemother. 2015 Aug; 59 (8):4956-61.
4. Farrell DJ, et al. Antimicrob Agents Chemother. 2017 Feb 23; 61 (3). pii: e02047-16.

Other Notes

Small volumes of GSK-2140944 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GSK-2140944 purchase

MBS3600308 is a biochemical targeting GSK-2140944.