BMS-823778 free base (BMS823778)

Name: BMS-823778 Free Base (BMS823778); MyBioSource
Brand: MyBioSource
SKU: MBS3600496
Price: 375 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3600496

BMS-823778 (BMS823778) is an orally available, potent and selective inhibitor of 11betaHSD-1 with IC50 of 2.3 nM. More details

$375 / 2 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

BMS-823778 free base, Biochemical

Full Product Name

BMS-823778 free base

Product Synonym Names

BMS823778

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

327.812

Target

11beta-HSD

Receptor

11beta-HSD

Chemical Name

2-(3-(1-(4-chlorophenyl)cyclopropyl)-[1, 2, 4]triazolo[4, 3-a]pyridin-8-yl)propan-2-ol

SMILES

CC(C)(C1=CC=CN2C1=NN=C2C3(CC3)C4=CC=C(C=C4)Cl)O

Molecular Formula

C18H18ClN3O

CAS Number

1140897-32-0

Product Categories/Family for BMS-823778 free base biochemical

Diabetes; Metabolic Enzyme/Protease; Metabolic Disease

Product References and Citations for BMS-823778 free base biochemical

1. Cheng Y, et al. Br J Clin Pharmacol. 2018 Jan; 84 (1):130-141.
2. Jun Li, et al. Discovery of Clinical Candidate BMS-823778 as an Inhibitor of Human 11beta-Hydroxysteroid Dehydrogenase Type 1 (11beta-HSD-1). ACS Med. Chem. Lett. 2018 Nov. DOI: 10.1021/acsmedchemlett.8b00307.

Other Notes

Small volumes of BMS-823778 free base biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for BMS-823778 free base purchase

MBS3600496 is a biochemical targeting BMS-823778 free base.