Ly 2456302 (CERC-501)

Name: Ly 2456302 (CERC-501); MyBioSource
Brand: MyBioSource
SKU: MBS3600590
Price: 235 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3600590

LY 2456302 (CERC-501, JSPA 0658, Aticaprant) is a potent, selective, short-acting antagonist of kappa-opioid receptor (KOR) with Ki of 0.81 nM. More details

$235 / 2 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

LY 2456302, Biochemical

Full Product Name

LY 2456302

Product Synonym Names

CERC-501; JSPA 0658; Aticaprant

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

418.512

Suitability

DMSO: >=100mg/mL (238.95mM)

Target

Opioid Receptor

Receptor

Opioid Receptor

Chemical Name

4-(4-(((2S)-2-(3, 5-dimethylphenyl)-1-pyrrolidinyl)methyl)phenoxy)-3-fluoro-benzamide

SMILES

O=C(N)C1=CC=C(OC2=CC=C(CN3[C@H](C4=CC(C)=CC(C)=C4)CCC3)C=C2)C(F)=C1

Molecular Formula

C26H27FN2O2

CAS Number

1174130-61-0

Product Categories/Family for LY 2456302 biochemical

Depression; Endocrinology/Hormones; Neurological Disease

Product References and Citations for LY 2456302 biochemical

1. Rorick-Kehn LM, et al. Neuropharmacology. 2014 Feb; 77:131-44.
2. Jackson KJ, et al. Neuropharmacology. 2015 Oct; 97:270-4.
3. Naganawa M, et al. J Pharmacol Exp Ther. 2016 Feb; 356 (2):260-6.

Other Notes

Small volumes of LY 2456302 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for LY 2456302 purchase

MBS3600590 is a biochemical targeting LY 2456302.