Lumateperone Tosylate (ITI-007)

Name: Lumateperone Tosylate (ITI-007); MyBioSource
Brand: MyBioSource
SKU: MBS3600638
Price: 235 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3600638

Lumateperone (ITI-007) is a potent 5-HT2A antagonist (Ki=0.54 nM), postsynaptic D2 antagonist(Ki=32 nM), and SERT blocker (Ki= 61 nM). More details

$235 / 5 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Lumateperone tosylate, Biochemical

Full Product Name

Lumateperone tosylate

Product Synonym Names

ITI-007

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

565.6987

Suitability

10mM in DMSO

Target

5-HT Receptor

Receptor

5-HT Receptor

Chemical Name

1-Butanone, 1-(4-fluorophenyl)-4-[(6bR, 10aS)-2, 3, 6b, 9, 10, 10a-hexahydro-3-methyl-1H-pyrido[3', 4':4, 5]pyrrolo[1, 2, 3-de]quinoxalin-8(7H)-yl]-, 4-methylbenzenesulfonate(1:1)

SMILES

CC1=CC=C(C=C1)S(=O)(=O)O.CN1CCN2C3CCN(CC3C4=C2C1=CC=C4)CCCC(=O)C5=CC=C(C=C5)F

Molecular Formula

C31H36FN3O4S

CAS Number

1187020-80-9

Product Categories/Family for Lumateperone tosylate biochemical

Schizophrenia; Endocrinology/Hormones; Neurological Disease

Product References and Citations for Lumateperone tosylate biochemical

1. Li P, et al. J Med Chem. 2014 Mar 27; 57 (6):2670-82.
2. Snyder GL, et al. Psychopharmacology (Berl). 2015 Feb; 232 (3):605-21.
3. Davis RE, et al. Psychopharmacology (Berl). 2015 Aug; 232 (15):2863-72.

Other Notes

Small volumes of Lumateperone tosylate biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Lumateperone tosylate purchase

MBS3600638 is a biochemical targeting Lumateperone tosylate.