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CX-6258

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3600741

A potent, selective, and orally efficacious pan-Pim inhibitor with IC50 of 5/25/16 nM for Pim1/2/3, respectively. More details

$255 / 5 mg +1 FREE 8GB USB
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
CX-6258, Biochemical
Full Product Name
CX-6258
Product Synonym Names
CX6258; CX 6258
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
461.9401
Suitability
10mM in DMSO
Target
Pim
Receptor
Pim1; Pim2; Pim3
Chemical Name
2H-Indol-2-one, 5-chloro-3-[[5-[3-[(hexahydro-4-methyl-1H-1, 4-diazepin-1-yl)carbonyl]phenyl]-2-furanyl]methylene]-1, 3-dihydro-, (3E)
SMILES
CN1CCCN(CC1)C(=O)C2=CC=CC(=C2)C3=CC=C(O3)/C=C/4C5=C(C=CC(=C5)Cl)NC4=O
Molecular Formula
C26H24ClN3O3
CAS Number
1202916-90-2

Product Categories/Family for CX-6258 biochemical

Blood cancer; JAK/STAT Signaling; Cancer

Structure of CX-6258 biochemical

Cx-6258 Biochemical – Cat# MBS3600741

Product References and Citations for CX-6258 biochemical

1. Haddach M, et al. ACS Med Chem Lett. 2011 Dec 27; 3 (2):135-9.
2. Padmanabhan A, et al. J Cell Biochem. 2013 May; 114 (5):1050-7.
3. Rebello RJ, et al. Clin Cancer Res. 2016 Nov 15; 22 (22):5539-5552.

Other Notes

Small volumes of CX-6258 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for CX-6258 purchase

MBS3600741 is a biochemical targeting CX-6258.
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