Sapanisertib (INK-128)

Name: Sapanisertib (INK-128); MyBioSource
Brand: MyBioSource
SKU: MBS3600859
Price: 235 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3600859

Sapanisertib (INK-128, MLN0128) is a potent, ATP-competitive, orally active dual mTORC1/2 inhibitor with Ki of 1.4 nM in cell-free assays. More details

$235 / 2 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Sapanisertib, Biochemical

Full Product Name

Sapanisertib

Product Synonym Names

INK-128; MLN0128

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

309.33

Suitability

10mM in DMSO

Target

mTOR

Receptor

mTOR; PI3Kalpha; PI3Kgamma; PI3Kdelta

Chemical Name

1H-Pyrazolo[3, 4-d]pyrimidin-4-amine, 3-(2-amino-5-benzoxazolyl)-1-(1-methylethyl)

SMILES

NC1=C2C(N(C(C)C)N=C2C3=CC=C(OC(N)=N4)C4=C3)=NC=N1

Molecular Formula

C15H15N7O

CAS Number

1224844-38-5

Product Categories/Family for Sapanisertib biochemical

Brain Cancer; PI3K/Akt/mTOR signaling; Cancer

Product References and Citations for Sapanisertib biochemical

1. Hsieh AC, et al. Nature. 2012 Feb 22; 485 (7396):55-61.
2. Gkmen-Polar Y, et al. Breast Cancer Res Treat.
3. Maiso P, et al. Blood. 2011 Dec 22; 118 (26):6860-70.
4. Janes MR, et al. Leukemia. 2013 Mar; 27 (3):586-94.

Other Notes

Small volumes of Sapanisertib biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Sapanisertib purchase

MBS3600859 is a biochemical targeting Sapanisertib.