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ETP-46321

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3601011

ETP-46321 is a potent, selective, orally bioavailable dual PI3K alpha/delta inhibitor with IC50 of 2.3/14.2 nM. More details

$255 / 5 mg +1 FREE 8GB USB
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
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Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
ETP-46321, Biochemical
Full Product Name
ETP-46321
Product Synonym Names
ETP 46321; ETP46321
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
473.5519
Suitability
DMSO: >=33mg/mL
Target
PI3K
Receptor
PI3K
Chemical Name
2-Pyrimidinamine, 5-[2-[[4-(methylsulfonyl)-1-piperazinyl]methyl]-8-(4-morpholinyl)imidazo[1, 2-a]pyrazin-6-yl]
SMILES
NC1=NC=C(C2=CN3C(C(N4CCOCC4)=N2)=NC(CN5CCN(S(=O)(C)=O)CC5)=C3)C=N1
Molecular Formula
C20H27N9O3S
CAS Number
1252594-99-2

Product Categories/Family for ETP-46321 biochemical

PI3K/Akt/mTOR signaling; Cancer

Structure of ETP-46321 biochemical

ETP-46321 Biochemical – Cat# MBS3601011

Product References and Citations for ETP-46321 biochemical

1. Marti­nez Gonzalez S, et al. Bioorg Med Chem Lett. 2012 May 15; 22 (10):3460-6.
2. Granda TG, et al. Invest New Drugs. 2013 Feb; 31 (1):66-76.
3. Aragoneses-Fenoll L, et al. Biochem Pharmacol. 2016 Apr 15; 106:56-69.

Other Notes

Small volumes of ETP-46321 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for ETP-46321 purchase

MBS3601011 is a biochemical targeting ETP-46321.
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