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I-BET151 (GSK1210151A)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3601204

MBS3601204 is a biochemical targeting I-BET151. I-BET151 (GSK1210151A) is a potent, selective BET bromodomain inhibitor. More details

$240 / 2 mg +1 FREE 8GB USB
Product Documentation
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Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
I-BET151, Biochemical
Full Product Name
I-BET151
Product Synonym Names
GSK1210151A; I-BET 151; GSK-1210151A
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
415.4445
Suitability
10mM in DMSO
Target
Bromodomain
Receptor
BRD2; BRD3; BRD4
Chemical Name
2H-Imidazo[4, 5-c]quinolin-2-one, 7-(3, 5-dimethyl-4-isoxazolyl)-1, 3-dihydro-8-methoxy-1-[(1R)-1-(2-pyridinyl)ethyl]
SMILES
O=C(N1[C@@H](C2=NC=CC=C2)C)NC3=C1C4=CC(OC)=C(C5=C(C)ON=C5C)C=C4N=C3
Molecular Formula
C23H21N5O3
CAS Number
1300031-49-5

Product Categories/Family for I-BET151 biochemical

Chromatin/Epigenetic; Cancer

Structure of I-BET151 biochemical

I-BET151 GSK1210151A Biochemical – Cat# MBS3601204

Product References and Citations for I-BET151 biochemical

1. Dawson MA, et al. Nature. 2011 Oct 2; 478 (7370):529-33.
2. Mirguet O, et al. Bioorg Med Chem Lett. 2012 Apr 15; 22 (8):2963-7.
3. Chaidos A, et al. Blood. 2014 Jan 30; 123 (5):697-705.
4. Wyspiańska BS, et al. Leukemia. 2014 Jan; 28 (1):88-97.

Other Notes

Small volumes of I-BET151 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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