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EPZ004777

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3601359

MBS3601359 is a biochemical targeting EPZ004777. EPZ004777 is a potent, selective DOT1L inhibitor with IC50 of 0.4 nM. More details

$255 / 5 mg +1 FREE 8GB USB
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
EPZ004777, Biochemical
Full Product Name
EPZ004777
Product Synonym Names
EPZ004777; EPZ 004777
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
539.67
Suitability
Ethanol: 100mg/mL (185.29mM)
DMSO: 100mg/mL (185.29mM)
Target
HMTase
Receptor
DOT1L
Chemical Name
1-(3-((((2R, 3S, 4R, 5R)-5-(4-amino-7H-pyrrolo[2, 3-d]pyrimidin-7-yl)-3, 4-dihydroxytetrahydrofuran-2-yl)methyl)(isopropyl)amino)propyl)-3-(4-(tert-butyl)phenyl)urea
SMILES
O=C(NC1=CC=C(C(C)(C)C)C=C1)NCCCN(C[C@H]2O[C@@H](N3C=CC4=C(N)N=CN=C43)[C@H](O)[C@@H]2O)C(C)C
Molecular Formula
C28H41N7O4
CAS Number
1338466-77-5

Product Categories/Family for EPZ004777 biochemical

Chromatin/Epigenetic; Cancer

Structure of EPZ004777 biochemical

EPZ004777 Biochemical – Cat# MBS3601359

Product References and Citations for EPZ004777 biochemical

1. Daigle SR, et al. Y Cell. 2011, 20 (1), 53-65.

Other Notes

Small volumes of EPZ004777 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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