GSK126 (GSK2816126)

Name: GSK126 (GSK2816126); MyBioSource
Brand: MyBioSource
SKU: MBS3601403
Price: 220 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3601403

GSK126 is a potent, highly selective EZH2 methyltransferase inhibitor with IC50 of 9.9 nM. More details

$220 / 2 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

GSK126, Biochemical

Full Product Name

GSK126

Product Synonym Names

GSK2816126; GSK-2816126; GSK 2816126

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

526.67

Suitability

DMSO: 3mg/mL warmed (5.69mM)

Target

HMTase

Receptor

EZH2

Chemical Name

(S)-1-(sec-butyl)-N-((4, 6-dimethyl-2-oxo-1, 2-dihydropyridin-3-yl)methyl)-3-methyl-6-(6-(piperazin-1-yl)pyridin-3-yl)-1H-indole-4-carboxamide

SMILES

O=C(C1=CC(C2=CC=C(N3CCNCC3)N=C2)=CC4=C1C(C)=CN4[C@@H](C)CC)NCC5=C(C)C=C(C)NC5=O

Molecular Formula

C31H38N6O2

CAS Number

1346574-57-9

Product Categories/Family for GSK126 biochemical

Chromatin/Epigenetic; Cancer

Product References and Citations for GSK126 biochemical

1.McCabe MT, et al. Nature. 2012, 492 (7427), 108-112.

Other Notes

Small volumes of GSK126 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GSK126 purchase

MBS3601403 is a biochemical targeting GSK126.