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GSK343

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3601407

GSK343 is a potent and selective EZH2 inhibitor with IC50 of 4 nM, showing 60 fold selectivity against EZH1. More details

$240 / 5 mg +1 FREE 8GB USB
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
GSK343, Biochemical
Full Product Name
GSK343
Product Synonym Names
GSK343; GSK-343; GSK 343
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
541.69
Suitability
Ethanol: 4mg/mL (7.38mM)
DMSO: 1mg/mL warmed (1.84mM)
Target
HMTase
Receptor
EZH1; EZH2
Chemical Name
1-isopropyl-N-((6-methyl-2-oxo-4-propyl-1, 2-dihydropyridin-3-yl)methyl)-6-(2-(4-methylpiperazin-1-yl)pyridin-4-yl)-1H-indazole-4-carboxamide.
SMILES
O=C(C1=CC(C2=CC(N3CCN(C)CC3)=NC=C2)=CC4=C1C=NN4C(C)C)NCC5=C(CCC)C=C(C)NC5=O
Molecular Formula
C31H39N7O2
CAS Number
1346704-33-3

Product Categories/Family for GSK343 biochemical

Chromatin/Epigenetic; Cancer

Structure of GSK343 biochemical

GSK343 Biochemical – Cat# MBS3601407

Product References and Citations for GSK343 biochemical

1.Verma SK, et al. ACS Med Chem Lett. 2012, 3, 1091-1096.

Other Notes

Small volumes of GSK343 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GSK343 purchase

MBS3601407 is a biochemical targeting GSK343.
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