Firuglipel (DS-8500)

Name: Firuglipel (DS-8500); MyBioSource
Brand: MyBioSource
SKU: MBS3601532
Price: 585 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3601532

Firuglipel (DS-8500, DS8500a) is a novel potent, selective, orally available GPR119 agonist with EC50 of 51.5 nM in human GPR119-expressing CHO-K1 cells. More details

$585 / 5 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Firuglipel, Biochemical

Full Product Name

Firuglipel

Product Synonym Names

DS-8500; DS8500a

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

467.497

Suitability

10mM in DMSO

Target

GPR119

Receptor

GPR119

Chemical Name

4-(5-{(1R)-1-[4-(cyclopropanecarbonyl)phenoxy]propyl}-1, 2, 4-oxadiazol-3-yl)-2-fluoro-N-[(2R)-1-hydroxypropan-2-yl]benzamide

SMILES

O=C(N[C@@H](C)CO)C1=CC=C(C2=NOC([C@@H](OC3=CC=C(C(C4CC4)=O)C=C3)CC)=N2)C=C1F

Molecular Formula

C25H26FN3O5

CAS Number

1371591-51-3

Product Categories/Family for Firuglipel biochemical

Diabetes; GPCR/G Protein; Metabolic Disease

Product References and Citations for Firuglipel biochemical

1. Patent WO2012050151.
2.Inagaki N, et al. BMJ Open Diabetes Res Care. 2017 Sep 29; 5 (1):e000424.
3.Terauchi Y, et al. J Diabetes Investig. 2018 Apr 1. doi: 10.1111/jdi.12846.
4.Makino C, et al. Xenobiotica. 2018 Aug 20:1-33. doi: 10.1080/00498254.2018.1514545.

Other Notes

Small volumes of Firuglipel biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Firuglipel purchase

MBS3601532 is a biochemical targeting Firuglipel.