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GLPG 0974

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3601618

GLPG 0974 is a potent, selective free fatty acid receptor 2 (FFA2, GPR43) antagonist with IC50 of 95 nM. More details

$290 / 5 mg +1 FREE 8GB USB
Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
GLPG 0974, Biochemical
Full Product Name
GLPG 0974
Product Synonym Names
GLPG0974
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
484.995
Target
FFAR
Receptor
FFAR
Chemical Name
4-[[[(2R)-1-(Benzo[b]thien-3-ylcarbonyl)-2-methyl-2-azetidinyl]carbonyl][(3-chlorophenyl)
SMILES
O=C(O)CCCN(C([C@]1(C)N(C(C2=CSC3=CC=CC=C23)=O)CC1)=O)CC4=CC=CC(Cl)=C4
Molecular Formula
C25H25ClN2O4S
CAS Number
1391076-61-1

Product Categories/Family for GLPG 0974 biochemical

Ulcer; GPCR/G Protein; Other Indications

Structure of GLPG 0974 biochemical

GLPG 0974 Biochemical – Cat# MBS3601618

Product References and Citations for GLPG 0974 biochemical

1. Pizzonero M, et al. J Med Chem. 2014 Dec 11; 57 (23):10044-57.
2. Sergeev E, et al. J Biol Chem. 2016 Jan 1; 291 (1):303-17.
3. Namour F, et al. Br J Clin Pharmacol. 2016 Jul; 82 (1):139-48.

Other Notes

Small volumes of GLPG 0974 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GLPG 0974 purchase

MBS3601618 is a biochemical targeting GLPG 0974.
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