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GCGR-IN-17 (PF-06291874)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3601636

MBS3601636 is a biochemical targeting GCGR-IN-17. A highly potent glucagon receptor antagonist with Ki of 14 nM for hGCGR. More details

$240 / 5 mg +1 FREE 8GB USB
Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
GCGR-IN-17, Biochemical
Full Product Name
GCGR-IN-17
Product Synonym Names
PF-06291874; PF06291874; PF-6291874
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
503.5134
Suitability
DMSO: >=30mg/mL
Target
Glucagon Receptor
Receptor
Glucagon Receptor
Chemical Name
glucagon receptor antagonists-4, N-[4-[(1S)-1-[3, 5-dimethyl-4-[4-(trifluoromethyl)-1H-pyrazol-1-yl]phenoxy]butyl]benzoyl]
SMILES
O=C(O)CCNC(C1=CC=C([C@@H](OC2=CC(C)=C(C(C)=C2)N3C=C(C=N3)C(F)(F)F)CCC)C=C1)=O
Molecular Formula
C26H28F3N3O4
CAS Number
1393124-08-7

Product Categories/Family for GCGR-IN-17 biochemical

Diabetes; GPCR/G Protein; Metabolic Disease

Structure of GCGR-IN-17 biochemical

GCGR-IN-17 PF-06291874 Biochemical – Cat# MBS3601636

Product References and Citations for GCGR-IN-17 biochemical

1. Guzman-Perez A, et la. Bioorg Med Chem Lett. 2013 May 15; 23 (10):3051-8.

Other Notes

Small volumes of GCGR-IN-17 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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