• Call +1.858.633.0165 or Fax +1.858.633.0166 or Contact Us

CCT-244747

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3601693

A novel, potent, highly selective, orally active, ATP competitive CHK1 inhibitor with biochemical IC50 of 8 nM; displays 75-fold selectivity against FLT3 and >1,000-fold selectivity against CHK2 and CDK1. More details

$405 / 10 mg +1 FREE 8GB USB
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
CCT-244747, Biochemical
Full Product Name
CCT-244747
Product Synonym Names
CCT 244747; CCT244747
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
408.457
Suitability
10mM in DMSO
Target
Chk
Receptor
Chk
Chemical Name
2-Pyrazinecarbonitrile, 3-[(1R)-2-(dimethylamino)-1-methylethoxy]-5-[[4-methoxy-5-(1-methyl-1H-pyrazol-4-yl)-2-pyridinyl]amino]
SMILES
N#CC1=NC=C(N=C1O[C@@H](CN(C)C)C)NC2=NC=C(C(OC)=C2)C3=CN(N=C3)C
Molecular Formula
C20H24N8O2
CAS Number
1404095-34-6

Product Categories/Family for CCT-244747 biochemical

Angiogenesis; Cancer

Structure of CCT-244747 biochemical

CCT-244747 Biochemical – Cat# MBS3601693

Product References and Citations for CCT-244747 biochemical

1. Walton MI, et al. Clin Cancer Res. 2012 Oct 15; 18 (20):5650-61.
2. Lainchbury M, et al. J Med Chem. 2012 Nov 26; 55 (22):10229-40.
3. Barker HE, et al. Mol Cancer Ther. 2016 Sep; 15 (9):2042-54.

Other Notes

Small volumes of CCT-244747 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for CCT-244747 purchase

MBS3601693 is a biochemical targeting CCT-244747.
Request a Quote

Please fill out the form below and our representative will get back to you shortly.

MBS000000
Contact Us

Please fill out the form below and our representative will get back to you shortly.

MBS000000