ACT-541468 (Nemorexant)

Name: ACT-541468 (Nemorexant); MyBioSource
Brand: MyBioSource
SKU: MBS3602099
Price: 1515 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3602099

A potent, selective, dual orexin receptor 1 and 2 (OX1 and OX2) antagonist with Kb of 0.52 and 0.78 nM, respectively. More details

$1515 / 5 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

ACT-541468, Biochemical

Full Product Name

ACT-541468

Product Synonym Names

Nemorexant; ACT541468; DORA

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

450.927

Suitability

DMSO: >=250mg/mL (554.42mM)

Target

Orexin Receptor

Receptor

Orexin Receptor

Chemical Name

(S)-(2-(5-chloro-4-methyl-1H-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1-yl)(5-methoxy-2-(2H-1, 2, 3-triazol-2-yl)phenyl)methanone

SMILES

O=C(N1[C@](C)(C2=NC3=C(C)C(Cl)=CC=C3N2)CCC1)C4=CC(OC)=CC=C4N5N=CC=N5

Molecular Formula

C23H23ClN6O2

CAS Number

1505484-82-1

Product Categories/Family for ACT-541468 biochemical

Sleep Disorder; GPCR/G Protein; Neurological Disease

Product References and Citations for ACT-541468 biochemical

1. Treiber A, et al. J Pharmacol Exp Ther. 2017 Sep; 362 (3):489-503.

Other Notes

Small volumes of ACT-541468 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for ACT-541468 purchase

MBS3602099 is a biochemical targeting ACT-541468.