Nalfurafine (TRK-820)

Name: Nalfurafine (TRK-820); MyBioSource
Brand: MyBioSource
SKU: MBS3602134
Price: 375 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3602134

Nalfurafine (TRK-820, TRK820) is potent, selective agonist of kappa-opioid receptor with Ki of 3.5 nM, 15-fold less potent for uOR and little affinity for deltaOR (Ki=53 and 1,200 nM, respectively). More details

$375 / 2 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Nalfurafine, Biochemical

Full Product Name

Nalfurafine

Product Synonym Names

TRK-820; TRK820

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

476.5641

Suitability

10mM in DMSO

Target

Opioid Receptor

Receptor

Opioid Receptor

Chemical Name

2-Propenamide, N-[(5alpha, 6beta)-17-(cyclopropylmethyl)-4, 5-epoxy-3, 14-dihydroxymorphinan-6-yl]-3-(3-furanyl)-N-methyl-, (2E)

SMILES

CN(C1CCC2(C3CC4=C5C2(C1OC5=C(C=C4)O)CCN3CC6CC6)O)C(=O)C=CC7=COC=C7

Molecular Formula

C28H32N2O5

CAS Number

152657-84-6

Product Categories/Family for Nalfurafine biochemical

Other Disease; Endocrinology/Hormones; Other Indications

Product References and Citations for Nalfurafine biochemical

1. Nagase H, et al. Chem Pharm Bull (Tokyo). 1998 Feb; 46 (2):366-9.
2. Seki T, et al. Eur J Pharmacol. 1999 Jul 2; 376 (1-2):159-67.
3. Endoh T, et al. Life Sci. 1999; 65 (16):1685-94.
4. Endoh T, et al. Eur J Pharmacol. 2000 Jan 10; 387 (2):133-40.

Other Notes

Small volumes of Nalfurafine biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Nalfurafine purchase

MBS3602134 is a biochemical targeting Nalfurafine.