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TGR-1202 R-enantiomer

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3602155

TGR-1202 R-enantiomer is is the less active enantiomer of TGR-1202 (Umbralisib), TGR-1202 is a potent, selective, orally available PI3Kdelta inhibitor with IC50 of 22 nM. More details

$540 / 5 mg +1 FREE 8GB USB
Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
TGR-1202 R-enantiomer, Biochemical
Full Product Name
TGR-1202 R-enantiomer
Product Synonym Names
RP5264 R-enantiomer; TGR1202 R-enantiomer
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
571.5492
Suitability
10mM in DMSO
Target
PI3K
Receptor
PI3K
Chemical Name
4H-1-Benzopyran-4-one, 2-[(1R)-1-[4-amino-3-[3-fluoro-4-(1-methylethoxy)phenyl]-1H-pyrazolo[3, 4-d]pyrimidin-1-yl]ethyl]-6-fluoro-3-(3-fluorophenyl)
SMILES
O=C1C(C2=CC=CC(F)=C2)=C([C@@H](C)N3N=C(C4=CC=C(OC(C)C)C(F)=C4)C5=C(N)N=CN=C53)OC6=CC=C(F)C=C16
Molecular Formula
C31H24F3N5O3
CAS Number
1532533-69-9

Product Categories/Family for TGR-1202 R-enantiomer biochemical

PI3K/Akt/mTOR signaling; Other Indications

Structure of TGR-1202 R-enantiomer biochemical

TGR-1202 R-enantiomer Biochemical – Cat# MBS3602155

Product References and Citations for TGR-1202 R-enantiomer biochemical

1. Locatelli SL, et al. Leukemia. 2016 Dec; 30 (12):2402-2405.
2. Deng C, et al. Blood. 2017 Jan 5; 129 (1):88-99.
3. Burris HA 3rd, et al. Lancet Oncol. 2018 Feb 20. pii: S1470-2045 (18)30082-2.
4. Lampson BL, et al. Expert Opin Investig Drugs. 2017 Nov; 26 (11):1267-1279.

Other Notes

Small volumes of TGR-1202 R-enantiomer biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for TGR-1202 R-enantiomer purchase

MBS3602155 is a biochemical targeting TGR-1202 R-enantiomer.
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