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EPZ-011989

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3602289

EPZ-011989 (EPZ011989) is a potent, selective, orally bioavailable inhibitor of EZH2 with Ki of < 3 nM. More details

$215 / 5 mg +1 FREE 8GB USB
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
EPZ-011989, Biochemical
Full Product Name
EPZ-011989
Product Synonym Names
EPZ011989
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
605.8105
Suitability
DMSO: >=33mg/mL
Target
HMTase
Receptor
EZH2
Chemical Name
Benzamide, N-[(1, 2-dihydro-4, 6-dimethyl-2-oxo-3-pyridinyl)methyl]-3-[ethyl[trans-4-[(2-methoxyethyl)methylamino]cyclohexyl]amino]-2-methyl-5-[3-(4-morpholinyl)-1-propyn-1-yl]
SMILES
O=C(NCC1=C(C)C=C(C)NC1=O)C2=CC(C#CCN3CCOCC3)=CC(N(CC)[C@H]4CC[C@H](N(CCOC)C)CC4)=C2C
Molecular Formula
C35H51N5O4
CAS Number
1598383-40-4

Product Categories/Family for EPZ-011989 biochemical

Blood cancer; Chromatin/Epigenetic; Cancer

Product References and Citations for EPZ-011989 biochemical

1. Campbell JE, et al. ACS Med Chem Lett. 2015 Mar 4; 6 (5):491-5.
2. Gardner EE, et al. Cancer Cell. 2017 Feb 13; 31 (2):286-299.

Other Notes

Small volumes of EPZ-011989 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for EPZ-011989 purchase

MBS3602289 is a biochemical targeting EPZ-011989.
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