• Call +1.858.633.0165 or Fax +1.858.633.0166 or Contact Us

GSK-481

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3602392

A highly potent, monokinase selective and ATP-competitive inhibitor of RIP1 kinase with biochemical IC50 of 10 nM. More details

$215 / 2 mg +1 FREE 8GB USB
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
GSK-481, Biochemical
Full Product Name
GSK-481
Product Synonym Names
GSK481; GSK481
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
377.3932
Suitability
DMSO: >=35mg/mL
Target
RIP kinase
Receptor
RIP1
Chemical Name
3-Isoxazolecarboxamide, 5-(phenylmethyl)-N-[(3S)-2, 3, 4, 5-tetrahydro-5-methyl-4-oxo-1, 5-benzoxazepin-3-yl]
SMILES
O=C(C1=NOC(CC2=CC=CC=C2)=C1)N[C@H]3COC4=CC=CC=C4N(C)C3=O
Molecular Formula
C21H19N3O4
CAS Number
1622849-58-4

Product Categories/Family for GSK-481 biochemical

Apoptosis; Cancer

Structure of GSK-481 biochemical

GSK-481 Biochemical – Cat# MBS3602392

Product References and Citations for GSK-481 biochemical

1. Harris PA, et al. J Med Chem. 2016 Mar 10; 59 (5):2163-78.

Other Notes

Small volumes of GSK-481 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GSK-481 purchase

MBS3602392 is a biochemical targeting GSK-481.
Request a Quote

Please fill out the form below and our representative will get back to you shortly.

MBS000000
Contact Us

Please fill out the form below and our representative will get back to you shortly.

MBS000000