Fezolinetant (ESN-364)

Name: Fezolinetant (ESN-364); MyBioSource
Brand: MyBioSource
SKU: MBS3602438
Price: 305 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3602438

A potent, selective, orally active neurokinin-3 receptor (NK3R) antagonist with pIC50/pKi of 7.7/7.6. More details

$305 / 5 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Fezolinetant, Biochemical

Full Product Name

Fezolinetant

Product Synonym Names

ESN-364; ESN 364

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

358.3954

Suitability

DMSO: >=50mg/mL (139.51mM)

Target

Neurokinin Receptor

Receptor

Neurokinin Receptor

Chemical Name

[(8R)-5, 6-Dihydro-8-methyl-3-(3-methyl-1, 2, 4-thiadiazol-5-yl)-1, 2, 4-triazolo[4, 3-a]pyrazin-7(8H)-yl](4-fluorophenyl)methanone

SMILES

O=C(C1=CC=C(F)C=C1)N2[C@H](C)C3=NN=C(C4=NC(C)=NS4)N3CC2

Molecular Formula

C16H15FN6OS

CAS Number

1629229-37-3

Product Categories/Family for Fezolinetant biochemical

Other Disease; GPCR/G Protein; Other Indications

Product References and Citations for Fezolinetant biochemical

1. Hoveyda HR, et al. ACS Med Chem Lett. 2015 May 19; 6 (7):736-40.
2. Fraser GL, et al. Endocrinology. 2015 Nov; 156 (11):4214-25.
3. Fraser GL, et al. J Clin Endocrinol Metab. 2016 Feb; 101 (2):417-26.

Other Notes

Small volumes of Fezolinetant biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Fezolinetant purchase

MBS3602438 is a biochemical targeting Fezolinetant.