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THIQ 40

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3602721

THIQ 40 (THIQ40) is a potent, orally available ERalpha antagonist and selective estrogen receptor degrader (SERD) with IC50 of 17 nM (ERalpha binding) and 30 nM (ERalpha transcription), IC50 of 0.9 nM (ERalpha degradation). More details

$875 / 5 mg +1 FREE 8GB USB
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
THIQ 40, Biochemical
Full Product Name
THIQ 40
Product Synonym Names
THIQ40
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
427.544
Target
Estrogen Receptor/ERR
Receptor
Estrogen Receptor/ERR
Chemical Name
(E)-3-(4-(6-Hydroxy-2-(4-isopropylphenyl)-1-methyl-1, 2, 3, 4-tetrahydroisoquinolin-1-yl)phenyl)acrylic Acid
SMILES
CC(C)C1=CC=C(C=C1)N2CCC3=C(C2(C)C4=CC=C(C=C4)C=CC(=O)O)C=CC(=C3)O
Molecular Formula
C28H29NO3
CAS Number
1799430-91-3

Product Categories/Family for THIQ 40 biochemical

Endocrinology/Hormones

Structure of THIQ 40 biochemical

THIQ 40 Biochemical – Cat# MBS3602721

Product References and Citations for THIQ 40 biochemical

1. Burks HE, et al. J Med Chem. 2017 Apr 13; 60 (7):2790-2818.

Other Notes

Small volumes of THIQ 40 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for THIQ 40 purchase

MBS3602721 is a biochemical targeting THIQ 40.
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