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EPZ-031686

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3602763

A potent, selective, small molecule SMYD3 inhibitor (Biochem IC50=3 nM; Cell IC50= 36 nM). More details

$375 / 5 mg +1 FREE 8GB USB
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
EPZ-031686, Biochemical
Full Product Name
EPZ-031686
Product Synonym Names
EPZ031686; EPZ 031686
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
591.0858
Suitability
DMSO: >=5.9mg/mL
Target
HMTase
Receptor
HMTase
Chemical Name
1H-Indole-5-carboxamide, 6-chloro-2, 3-dihydro-2-oxo-N-[(3-endo)-8-[[[1-(4, 4, 4-trifluorobutyl)-4-piperidinyl]methyl]sulfonyl]-8-azabicyclo[3.2.1]oct-3-yl]
SMILES
O=C(C1=CC2=C(NC(C2)=O)C=C1Cl)N[C@H]3C[C@@](N4S(=O)(CC5CCN(CCCC(F)(F)F)CC5)=O)([H])CC[C@@]4([H])C3
Molecular Formula
C26H34ClF3N4O4S
CAS Number
1808011-22-4

Product Categories/Family for EPZ-031686 biochemical

Chromatin/Epigenetic; Cancer

Structure of EPZ-031686 biochemical

EPZ-031686 Biochemical – Cat# MBS3602763

Product References and Citations for EPZ-031686 biochemical

1. Mitchell LH, et al. ACS Med Chem Lett. 2015 Aug 27; 7 (2):134-8.
2. Rajajeyabalachandran G, et al. Expert Opin Ther Targets. 2017 Feb; 21 (2):145-157.

Other Notes

Small volumes of EPZ-031686 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for EPZ-031686 purchase

MBS3602763 is a biochemical targeting EPZ-031686.
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