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CCG-215022

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3602785

CCG-215022 (CCG215022) is a potent and selective pan GRK inhibitor with IC50 of 0.15/0.38/3.9 uM for GRK2/5/1 respectively. More details

$290 / 5 mg +1 FREE 8GB USB
Product Documentation
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Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
CCG-215022, Biochemical
Full Product Name
CCG-215022
Product Synonym Names
CCG215022; CCG 215022
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
499.4964
Suitability
DMSO: >=28mg/mL
Target
GRK (GPCRK)
Receptor
GRK1; GRK2; GRK5; PKA
Chemical Name
4-(4-fluoro-3-((pyridin-2-ylmethyl)carbamoyl)phenyl)-N-(1H-indazol-5-yl)-6-methyl-2-oxo-1, 2, 3, 4-tetrahydropyrimidine-5-carboxamide
SMILES
O=C(C1=C(F)C=CC(C2C(C(NC3=CC=C(NN=C4)C4=C3)=O)=C(C)NC(N2)=O)=C1)NCC5=NC=CC=C5
Molecular Formula
C26H22FN7O3
CAS Number
1813527-81-9

Product Categories/Family for CCG-215022 biochemical

Cancer

Structure of CCG-215022 biochemical

CCG-215022 Biochemical – Cat# MBS3602785

Product References and Citations for CCG-215022 biochemical

1. Homan KT, et al. J Biol Chem. 2015 Aug 21; 290 (34):20649-59.

Other Notes

Small volumes of CCG-215022 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for CCG-215022 purchase

MBS3602785 is a biochemical targeting CCG-215022.
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