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ACT 709478

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3602840

ACT 709478 is a potent, selective, orally-bioavailable, brain penetrant T-type calcium channel blocker with IC50 of 6.4, 18, and 7.5 nM for Cav3.1, Cav3.2, and Cav3.3 channels respectively. More details

$260 / 2 mg +1 FREE 8GB USB
Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
ACT 709478, Biochemical
Full Product Name
ACT 709478
Product Synonym Names
ACT709478
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
425.415
Suitability
DMSO: >=125mg/mL (293.83mM)
Target
Calcium Channel
Receptor
Calcium Channel
Chemical Name
N-(1-((5-Cyanopyridin-2-yl)methyl)-1H-pyrazol-3-yl)-2-(4-(1-(trifluoromethyl)cyclopropyl)-phenyl)acetamide
SMILES
O=C(NC1=NN(CC2=NC=C(C#N)C=C2)C=C1)CC3=CC=C(C4(C(F)(F)F)CC4)C=C3
Molecular Formula
C22H18F3N5O
CAS Number
1838651-58-3

Product Categories/Family for ACT 709478 biochemical

Epilepsy; GPCR/G Protein; Neurological Disease

Structure of ACT 709478 biochemical

ACT 709478 Biochemical – Cat# MBS3602840

Product References and Citations for ACT 709478 biochemical

1. Bezenon O, et al. J Med Chem. 2017 Nov 8. doi: 10.1021/acs.jmedchem.7b01236.

Other Notes

Small volumes of ACT 709478 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for ACT 709478 purchase

MBS3602840 is a biochemical targeting ACT 709478.
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