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GSK-6853

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3602992

A potent, highly selective and cell-active BRPF1 bromodomain inhibitor with TR-FRET pIC50 of 8.1. More details

$215 / 1mL*10mM (in DMSO) +1 FREE 8GB USB
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
GSK-6853, Biochemical
Full Product Name
GSK-6853
Product Synonym Names
GSK6853
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
409.4815
Suitability
DMSO: >=29mg/mL
Target
Bromodomain
Receptor
BRPF1; BRPF2; BRPF3
Chemical Name
Benzamide, N-[2, 3-dihydro-1, 3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxy
SMILES
O=C(NC1=C(N2[C@H](C)CNCC2)C=C(N3C)C(N(C)C3=O)=C1)C4=CC=CC=C4OC
Molecular Formula
C22H27N5O3
CAS Number
1910124-24-1

Product Categories/Family for GSK-6853 biochemical

Chromatin/Epigenetic; Cancer

Structure of GSK-6853 biochemical

GSK-6853 Biochemical – Cat# MBS3602992

Product References and Citations for GSK-6853 biochemical

1. Bamborough P, et al. ACS Med Chem Lett. 2016 May 9; 7 (6):552-7.

Other Notes

Small volumes of GSK-6853 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GSK-6853 purchase

MBS3602992 is a biochemical targeting GSK-6853.
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