OTX015 (HY-15743)

Name: OTX015 (HY-15743); MyBioSource
Brand: MyBioSource
SKU: MBS3603154
Price: 220 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3603154

OTX015 is a potent BET bromodomain inhibitor with EC50 ranging from 10 to 19 nM for BRD2, BRD3, and BRD4. Phase 1. More details

$220 / 2 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

OTX015, Biochemical

Full Product Name

OTX015

Product Synonym Names

HY-15743; ()-OTX015

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

491.99

Suitability

DMSO: 98mg/mL (199.19mM)
Ethanol: 98mg/mL (199.19mM)
Water: <1mg/mL (<1mM)

Target

Epigenetic Reader Domain

Receptor

BRDs

Chemical Name

(S)-2-(4-(4-chlorophenyl)-2, 3, 9-trimethyl-6H-thieno[3, 2-f][1, 2, 4]triazolo[4, 3-a][1, 4]diazepin-6-yl)-N-(4-hydroxyphenyl)acetamide.

SMILES

O=C(NC1=CC=C(O)C=C1)C[C@H]2C3=NN=C(C)N3C4=C(C(C)=C(C)S4)C(C5=CC=C(Cl)C=C5)=N2

Molecular Formula

C25H22ClN5O2S

CAS Number

202590-98-5

Product Categories/Family for OTX015 biochemical

Chromatin/Epigenetic; Cancer

Product References and Citations for OTX015 biochemical

1.Noel JK, et al. Mol Cancer Ther. 2013, 12, C244.

Other Notes

Small volumes of OTX015 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for OTX015 purchase

MBS3603154 is a biochemical targeting OTX015.