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GSK4027

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3603238

GSK4027 (GSK 4027, GSK-4027) is a potent, selective, cell-penetrant chemical probe of PCAF/GCN5 bromodomain with pKi of 8.9 for both. More details

$2445 / 5 mg +3 FREE 8GB USB
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
GSK4027, Biochemical
Full Product Name
GSK4027
Product Synonym Names
GSK 4027; GSK-4027
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
377.286
Suitability
DMSO: 50mg/mL (132.53mM)
Target
Bromodomain
Receptor
Bromodomain
Chemical Name
4-Bromo-2-methyl-5-(((3R, 5R)-1-methyl-5-phenylpiperidin-3-yl)amino)pyridazin-3(2H)-one
SMILES
CN1C[C@@H](C2=CC=CC=C2)C[C@@H](NC3=C(Br)C(N(C)N=C3)=O)C1
Molecular Formula
C17H21BrN4O
CAS Number
2079896-25-4

Product Categories/Family for GSK4027 biochemical

Chromatin/Epigenetic; Inflammation/Immunology

Structure of GSK4027 biochemical

GSK4027 Biochemical – Cat# MBS3603238

Product References and Citations for GSK4027 biochemical

1. Humphreys PG, et al. J Med Chem. 2017 Jan 26; 60 (2):695-709.

Other Notes

Small volumes of GSK4027 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GSK4027 purchase

MBS3603238 is a biochemical targeting GSK4027.
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