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ARQ-531

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3603293

ARQ-531 (ARQ531) is a potent, reversible, orally available inhibitor of both wild type and C481S-mutant BTK kinase with IC50 of 0.85 and 0.39 nM, respectively. More details

$220 / 2 mg +1 FREE 8GB USB
Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
ARQ-531, Biochemical
Full Product Name
ARQ-531
Product Synonym Names
ARQ531
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
478.933
Suitability
DMSO: >=50mg/mL (104.40mM)
Target
BTK
Receptor
BTK
Chemical Name
(2-chloro-4-phenoxyphenyl)(4-(((3R, 6S)-6-(hydroxymethyl)tetrahydro-2H-pyran-3-yl)amino)-7H-pyrrolo[2, 3-d]pyrimidin-5-yl)methanone
SMILES
O=C(C1=CC=C(OC2=CC=CC=C2)C=C1Cl)C3=CNC4=NC=NC(N[C@H]5CO[C@H](CO)CC5)=C43
Molecular Formula
C25H23ClN4O4
CAS Number
2095393-15-8

Product Categories/Family for ARQ-531 biochemical

Blood cancer; Tyrosine Kinase; Cancer

Structure of ARQ-531 biochemical

ARQ-531 Biochemical – Cat# MBS3603293

Product References and Citations for ARQ-531 biochemical

1. Reiff SD, et al. Cancer Discov. 2018 Aug 9. pii: CD-17-1409. doi: 10.1158/2159-8290.CD-17-1409.

Other Notes

Small volumes of ARQ-531 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for ARQ-531 purchase

MBS3603293 is a biochemical targeting ARQ-531.
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