Conivaptan (YM-087)

Name: Conivaptan (YM-087); MyBioSource
Brand: MyBioSource
SKU: MBS3603330
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3603330

A potent, selective, nonpeptide vasopressin V1A and V2 receptor antagonist with Ki of 0.48 nM and 3.04 nM respectively; has less potency for OT receptors and no effect on V1B receptor. More details

Please Inquire

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Conivaptan, Biochemical

Full Product Name

Conivaptan

Product Synonym Names

YM-087; ZINC 12503187

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

498.583

Target

Vasopressin Receptor

Receptor

Vasopressin Receptor

Chemical Name

N-[4-[(4, 5-Dihydro-2-methylimidazo[4, 5-d][1]benzazepin-6(1H)-yl)carbonyl]phenyl]-[1, 1'-Biphenyl]-2-carboxamide

SMILES

CC1=NC2=C(N1)CCN(C3=CC=CC=C32)C(=O)C4=CC=C(C=C4)NC(=O)C5=CC=CC=C5C6=CC=CC=C6

Molecular Formula

C32H26N4O2

CAS Number

210101-16-9

Product Categories/Family for Conivaptan biochemical

Other Disease; GPCR/G Protein; Other Indications

Product References and Citations for Conivaptan biochemical

1. Tahara A, et al. J Pharmacol Exp Ther. 1997 Jul; 282 (1):301-8.
2. Tahara A, et al. Cardiovasc Res. 1998 Apr; 38 (1):198-205.
3. Nakayama S, et al. Neurocrit Care. 2016 Apr; 24 (2):273-82.

Other Notes

Small volumes of Conivaptan biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Conivaptan purchase

MBS3603330 is a biochemical targeting Conivaptan.