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GNE-886

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3603340

GNE-886 is a potent and selective CECR2 bromodomain inhibitor with IC50 of 16 nM; shows a wide selectivity over the 40 bromodomains. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
GNE-886, Biochemical
Full Product Name
GNE-886
Product Synonym Names
GNE886
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
498.587
Target
Bromodomain
Receptor
Bromodomain
Chemical Name
6-allyl-N-(1-(6-(3-methoxyphenyl)pyrimidin-4-yl)piperidin-4-yl)-N-methyl-7-oxo-6, 7-dihydro-1H-pyrrolo[2, 3-c]pyridine-4-carboxamide
SMILES
CN(C1CCN(CC1)C2=NC=NC(=C2)C3=CC(=CC=C3)OC)C(=O)C4=CN(C(=O)C5=C4C=CN5)CC=C
Molecular Formula
C28H30N6O3
CAS Number
2101957-05-3

Product Categories/Family for GNE-886 biochemical

Chromatin/Epigenetic; Other Indications

Structure of GNE-886 biochemical

GNE-886 Biochemical – Cat# MBS3603340

Product References and Citations for GNE-886 biochemical

1. Crawford TD, et al. ACS Med Chem Lett. 2017 Jun 1; 8 (7):737-741.

Other Notes

Small volumes of GNE-886 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GNE-886 purchase

MBS3603340 is a biochemical targeting GNE-886.
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