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BETd-246

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3603420

A potent, second-generation BET protein degrader that exhibits superior selectivity, potency and antitumor activity. More details

$565 / 5 mg +1 FREE 8GB USB
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
BETd-246, Biochemical
Full Product Name
BETd-246
Product Synonym Names
BETd 246; BETd246
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
946.035
Suitability
DMSO: 200mg/mL (211.41mM)
Target
PROTAC
Receptor
PROTAC
Chemical Name
4-((3-cyclopropyl-1-ethyl-1H-pyrazol-5-yl)amino)-7-(3, 5-dimethylisoxazol-4-yl)-N-(3-(2-(2-(3-((2-(2, 6-dioxopiperidin-3-yl)-1, 3-dioxoisoindolin-4-yl)amino)propoxy)ethoxy)ethoxy)propyl)-6-methoxy-9H-pyrimido[4, 5-b]indole-2-carboxamide
SMILES
CCN1C(=CC(=N1)C2CC2)NC3=NC(=NC4=C3C5=CC(=C(C=C5N4)C6=C(ON=C6C)C)OC)C(=O)NCCCOCCOCCOCCCNC7=CC=CC8=C7C(=O)N(C8=O)C9CCC(=O)NC9=O
Molecular Formula
C48H55N11O10
CAS Number
2140289-17-2

Product Categories/Family for BETd-246 biochemical

PROTACs

Structure of BETd-246 biochemical

Betd-246 Biochemical – Cat# MBS3603420

Product References and Citations for BETd-246 biochemical

1. Bai L, et al. Cancer Res. 2017 May 1; 77 (9):2476-2487.

Other Notes

Small volumes of BETd-246 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for BETd-246 purchase

MBS3603420 is a biochemical targeting BETd-246.
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