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Dual DDR1 and DDR2 inhibitor 5n

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3603593

Dual DDR1 and DDR2 inhibitor 5n is a highly potent, selective, dual Discoidin domain receptor DDR1 and DDR2 inhibitor with Kd of 7.9 and 8.0 nM, IC50 of 9.4 and 20.4 nM, repectively. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Product Name
Dual DDR1 and DDR2 inhibitor 5n, Biochemical
Full Product Name
Dual DDR1 and DDR2 inhibitor 5n
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
560.625
Target
DDR
Receptor
DDR
Chemical Name
3-(Imidazo[1, 2-a]pyrazin-3-ylethynyl)-4-isopropyl-N-(3-((4-methylpiperazin-1-yl)methyl)-5-(trifluoromethyl)phenyl)benzamide
SMILES
CC(C)C1=C(C=C(C=C1)C(=O)NC2=CC(=CC(=C2)C(F)(F)F)CN3CCN(CC3)C)C#CC4=CN=C5N4C=CN=C5
Molecular Formula
C31H31F3N6O
CAS Number
2241813-33-0

Product Categories/Family for Dual DDR1 and DDR2 inhibitor 5n biochemical

Tyrosine Kinase

Structure of Dual DDR1 and DDR2 inhibitor 5n biochemical

Dual DDR1 and DDR2 Inhibitor 5n Biochemical – Cat# MBS3603593

Product References and Citations for Dual DDR1 and DDR2 inhibitor 5n biochemical

1. Wang Z, et al. J Med Chem. 2018 Aug 3. doi: 10.1021/acs.jmedchem.8b01045.

Other Notes

Small volumes of Dual DDR1 and DDR2 inhibitor 5n biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Dual DDR1 and DDR2 inhibitor 5n purchase

MBS3603593 is a biochemical targeting Dual DDR1 and DDR2 inhibitor 5n.
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