Pelitinib (EKB-569)

Name: Pelitinib (EKB-569); MyBioSource
Brand: MyBioSource
SKU: MBS3603778
Price: 235 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3603778

A potent, selective, orally active, irreversible inhibitor of EGFR with IC50 of 80 nM. More details

$235 / 5 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Pelitinib, Biochemical

Full Product Name

Pelitinib

Product Synonym Names

EKB-569; WAY-EKB 569; EKB569; EKB 569

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

467.9231

Suitability

DMSO: 16mg/mL

Target

EGFR

Receptor

EGFR; HER2/ErbB2; MEK; Raf; Src

Chemical Name

2-Butenamide, N-[4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-, (2E)

SMILES

O=C(NC1=C(OCC)C=C2N=CC(C#N)=C(NC3=CC=C(F)C(Cl)=C3)C2=C1)/C=C/CN(C)C

Molecular Formula

C24H23ClFN5O2

CAS Number

257933-82-7

Product Categories/Family for Pelitinib biochemical

Lung Cancer; Angiogenesis; Cancer

Product References and Citations for Pelitinib biochemical

1. Wissner A, et al. J Med Chem. 2003 Jan 2; 46 (1):49-63.
2. Nunes M, et al. Mol Cancer Ther. 2004 Jan; 3 (1):21-7.
3. Torrance CJ, et al. Nat Med. 2000 Sep; 6 (9):1024-8.

Other Notes

Small volumes of Pelitinib biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Pelitinib purchase

MBS3603778 is a biochemical targeting Pelitinib.