Sufugolix (TAK013)

Name: Sufugolix (TAK013); MyBioSource
Brand: MyBioSource
SKU: MBS3603985
Price: 235 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3603985

Sufugolix (TAK-013) is a highly potent and orally bioavailable non-peptide antagonist of luteinizing hormone-releasing hormone (LHRH) receptor with binding and functional IC50 of 0.1 and 0.06 nM for human LHRH, respectively. More details

$235 / 2 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Sufugolix, Biochemical

Full Product Name

Sufugolix

Product Synonym Names

TAK013; TAK-013; TAK 013

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

667.7242

Suitability

10mM in DMSO

Target

LHR

Receptor

humanLHRH; monkeyLHRH

Chemical Name

Urea, N-[4-[1-[(2, 6-difluorophenyl)methyl]-1, 2, 3, 4-tetrahydro-5-[[methyl(phenylmethyl)amino]methyl]-2, 4-dioxo-3-phenylthieno[2, 3-d]pyrimidin-6-yl]phenyl]-N'-methoxy

SMILES

O=C(NOC)NC1=CC=C(C(S2)=C(CN(C)CC3=CC=CC=C3)C(C(N4C5=CC=CC=C5)=O)=C2N(CC6=C(F)C=CC=C6F)C4=O)C=C1

Molecular Formula

C36H31F2N5O4S

CAS Number

308831-61-0

Product Categories/Family for Sufugolix biochemical

Other Disease; GPCR/G Protein; Other Indications

Product References and Citations for Sufugolix biochemical

1. Sasaki S, et al. J Med Chem. 2003 Jan 2; 46 (1):113-24.

Other Notes

Small volumes of Sufugolix biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Sufugolix purchase

MBS3603985 is a biochemical targeting Sufugolix.