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Darapladib (SB-480848)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3604218

MBS3604218 is a biochemical targeting Darapladib. A potent Lp-PLA2 inhibitor with IC50 of 0.25 nM. More details

$235 / 2 mg +1 FREE 8GB USB
Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
Darapladib, Biochemical
Full Product Name
Darapladib
Product Synonym Names
SB-480848; SB480848; SB 480848
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
666.7711
Suitability
10mM in DMSO
Target
Phospholipase
Receptor
Lp-PLA2
Chemical Name
1H-Cyclopentapyrimidine-1-acetamide, N-[2-(diethylamino)ethyl]-2-[[(4-fluorophenyl)methyl]thio]-4, 5, 6, 7-tetrahydro-4-oxo-N-[[4'-(trifluoromethyl)[1, 1'-biphenyl]-4-yl]methyl]
SMILES
O=C(N(CCN(CC)CC)CC1=CC=C(C2=CC=C(C(F)(F)F)C=C2)C=C1)CN(C3=C4CCC3)C(SCC5=CC=C(F)C=C5)=NC4=O
Molecular Formula
C36H38F4N4O2S
CAS Number
356057-34-6

Product Categories/Family for Darapladib biochemical

Atherosclerosis; Metabolic Enzyme/Protease; Cardiovascular Disease

Structure of Darapladib biochemical

Darapladib SB-480848 Biochemical – Cat# MBS3604218

Product References and Citations for Darapladib biochemical

1. Blackie JA, et al. Bioorg Med Chem Lett. 2003 Mar 24; 13 (6):1067-70.
2. Wilensky RL, et al. Nat Med. 2008 Oct; 14 (10):1059-66.
3. Serruys PW, et al. Circulation. 2008 Sep 9; 118 (11):1172-82.

Other Notes

Small volumes of Darapladib biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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