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Atopaxar hydrobromide

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3604575

A potent, reversible PAR-1 antagonist with IC50 of 19 nM; shows potent inhibitory effects on human platelet aggregation induced by thrombin and TRAP with IC50 of 64 nM and 31 nM, respectively. More details

$455 / 2 mg +1 FREE 8GB USB
Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
Atopaxar hydrobromide, Biochemical
Full Product Name
Atopaxar hydrobromide
Product Synonym Names
E5555 hydrobromide
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
608.54
Suitability
DMSO: 10mM (<1mg/mL refers to the product slightly soluble or insoluble)
Target
PAR
Receptor
PAR-1
Chemical Name
2-(5, 6-Diethoxy-7-fluoro-1, 3-dihydro-1-imino-2H-isoindol-2-yl)-1-[3-(1, 1-dimethylethyl)-4-methoxy-5-(4-morpholinyl)phenyl]ethanone hydrobromide
SMILES
COC1=C(N2CCOCC2)C=C(C(CN(CC3=C4C(F)=C(OCC)C(OCC)=C3)C4=N)=O)C=C1C(C)(C)C.[H]Br
Molecular Formula
C29H38FN3O5.HBr
CAS Number
474550-69-1

Product Categories/Family for Atopaxar hydrobromide biochemical

Thrombosis; GPCR/G Protein; Cardiovascular Disease

Structure of Atopaxar hydrobromide biochemical

Atopaxar Hydrobromide Biochemical – Cat# MBS3604575

Product References and Citations for Atopaxar hydrobromide biochemical

1. Serebruany VL, et al. Thromb Haemost. 2009 Jul; 102 (1):111-9.
2. Angiolillo DJ, et al. Eur Heart J. 2010 Jan; 31 (1):17-28.
3. Kogushi M, et al. Eur J Pharmacol. 2011 Apr 25; 657 (1-3):131-7.

Other Notes

Small volumes of Atopaxar hydrobromide biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Atopaxar hydrobromide purchase

MBS3604575 is a biochemical targeting Atopaxar hydrobromide.
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