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PHA-665752

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3604590

PHA-665752 is a potent, selective, ATP-competitive c-Met inhibitor with Ki/IC50 of 4/9 nM. More details

$240 / 5 mg +1 FREE 8GB USB
Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
PHA-665752, Biochemical
Full Product Name
PHA-665752
Product Synonym Names
PHA 665752; PHA665752
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
641.6078
Suitability
10mM in DMSO
Target
c-Met/HGFR
Receptor
c-Abl; c-Met; FGFR1; Flk1; RON
Chemical Name
2H-Indol-2-one, 5-[[(2, 6-dichlorophenyl)methyl]sulfonyl]-3-[[3, 5-dimethyl-4-[[(2R)-2-(1-pyrrolidinylmethyl)-1-pyrrolidinyl]carbonyl]-1H-pyrrol-2-yl]methylene]-1, 3-dihydro-, (3Z)
SMILES
O=C1NC2=C(C=C(S(=O)(CC3=C(Cl)C=CC=C3Cl)=O)C=C2)/C1=C/C4=C(C)C(C(N5[C@@H](CN6CCCC6)CCC5)=O)=C(C)N4
Molecular Formula
C32H34Cl2N4O4S
CAS Number
477575-56-7

Product Categories/Family for PHA-665752 biochemical

Angiogenesis; Cancer

Structure of PHA-665752 biochemical

PHA-665752 Biochemical – Cat# MBS3604590

Product References and Citations for PHA-665752 biochemical

1. Smolen GA, et al. Proc Natl Acad Sci U S A. 2006 Feb 14; 103 (7):2316-21.
2. Ma PC, et al. Clin Cancer Res. 2005 Mar 15; 11 (6):2312-9.
3. Hov H, et al. Clin Cancer Res. 2004 Oct 1; 10 (19):6686-94.
4. Christensen JG, et al. Cancer Res. 2003 Nov 1; 63 (21):7345-55.

Other Notes

Small volumes of PHA-665752 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for PHA-665752 purchase

MBS3604590 is a biochemical targeting PHA-665752.
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