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SB-705498

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3604692

A potent, selective and orally bioavailable TRPV1 antagonist with pKi of 7.6 (inhibition of capsaicin-mediated activation of hTRPV1 receptor). More details

$220 / 5 mg +1 FREE 8GB USB
Product Documentation
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Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
SB-705498, Biochemical
Full Product Name
SB-705498
Product Synonym Names
SB 705498; SB705498
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
429.2343
Suitability
10mM in DMSO
Target
TRP/TRPV Channel
Receptor
hTRPV1
Chemical Name
Urea, N-(2-bromophenyl)-N'-[(3R)-1-[5-(trifluoromethyl)-2-pyridinyl]-3-pyrrolidinyl]
SMILES
O=C(N[C@H]1CN(C2=NC=C(C(F)(F)F)C=C2)CC1)NC3=CC=CC=C3Br
Molecular Formula
C17H16BrF3N4O
CAS Number
501951-42-4

Product Categories/Family for SB-705498 biochemical

Pain; Membrane Transporter/Ion Channel; Neurological Disease

Structure of SB-705498 biochemical

Sb-705498 Biochemical – Cat# MBS3604692

Product References and Citations for SB-705498 biochemical

1. Rami HK, et al. Bioorg Med Chem Lett. 2006 Jun 15; 16 (12):3287-91.
2. Gunthorpe MJ, et al. J Pharmacol Exp Ther. 2007 Jun; 321 (3):1183-92.
3. Chizh BA, et al. Pain. 2007 Nov; 132 (1-2):132-41.

Other Notes

Small volumes of SB-705498 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for SB-705498 purchase

MBS3604692 is a biochemical targeting SB-705498.
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