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AMG-517

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3605508

AMG 517 is a potent and selective TRPV1 antagonist, antagonizes capsaicin, proton, and heat activation of TRPV1 with IC50 of 0.76 nM, 0.62 nM and 1.3 nM. More details

$235 / 5 mg +1 FREE 8GB USB
Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
AMG-517, Biochemical
Full Product Name
AMG-517
Product Synonym Names
AMG-517; AMG 517; AMG517; BD-0082
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
430.4
Suitability
DMSO: 86mg/mL (199.81mM)
Ethanol: <1mg/mL (<1mM)
Water: <1mg/mL (<1mM)
Target
TRP/TRPV Channel
Receptor
TRPV1
Chemical Name
Acetamide, N-(4-((6-(4-(trifluoromethyl)phenyl)-4-pyrimidinyl)oxy)-2-benzothiazolyl)
SMILES
CC(NC1=NC2=C(OC3=NC=NC(C4=CC=C(C(F)(F)F)C=C4)=C3)C=CC=C2S1)=O
Molecular Formula
C20H13F3N4O2S
CAS Number
659730-32-2

Product Categories/Family for AMG-517 biochemical

Membrane Transporter/Ion Channel; Neurological Disease

Structure of AMG-517 biochemical

AMG-517 Biochemical – Cat# MBS3605508

Product References and Citations for AMG-517 biochemical

1. Gavva NR, et al. J Pharmacol Exp Ther, 2007, 323 (1), 128-137.

Other Notes

Small volumes of AMG-517 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for AMG-517 purchase

MBS3605508 is a biochemical targeting AMG-517.
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