Linagliptin (BI 1356)

Name: Linagliptin (BI 1356); MyBioSource
Brand: MyBioSource
SKU: MBS3605550
Price: 220 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3605550

A highly potent, selective, long-acting, and orally bioavailable DPP-4 inhibitor with IC50 of 1 nM. More details

$220 / 50 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Linagliptin, Biochemical

Full Product Name

Linagliptin

Product Synonym Names

BI 1356; BI-1356; BI1356

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

472.5422

Suitability

10mM in DMSO

Target

DPP

Receptor

DPP-4

Chemical Name

1H-Purine-2, 6-dione, 8-[(3R)-3-amino-1-piperidinyl]-7-(2-butyn-1-yl)-3, 7-dihydro-3-methyl-1-[(4-methyl-2-quinazolinyl)methyl]

SMILES

O=C(N1CC2=NC(C)=C3C=CC=CC3=N2)N(C)C4=C(N(CC#CC)C(N5C[C@H](N)CCC5)=N4)C1=O

Molecular Formula

C25H28N8O2

CAS Number

668270-12-0

Product Categories/Family for Linagliptin biochemical

Diabetes; Metabolic Enzyme/Protease; Metabolic Disease

Product References and Citations for Linagliptin biochemical

1. Eckhardt M, et al. J Med Chem. 2007 Dec 27; 50 (26):6450-3.
2. Thomas L, et al. J Pharmacol Exp Ther. 2008 Apr; 325 (1):175-82.
3. Thomas L, et al. J Pharmacol Exp Ther. 2009 Feb; 328 (2):556-63.

Other Notes

Small volumes of Linagliptin biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Linagliptin purchase

MBS3605550 is a biochemical targeting Linagliptin.