BX795

Name: BX795; MyBioSource
Brand: MyBioSource
SKU: MBS3605694
Price: 240 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3605694

BX795 is a potent and relatively specific PDK1 inhibitor with IC50 of 6 nM; also inhibits TBK1 and IKKepsilon with IC50 of 6 nM and 41 nM. More details

$240 / 5 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

BX795, Biochemical

Full Product Name

BX795

Product Synonym Names

BX 795; BX-795

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

591.4677

Suitability

10mM in DMSO

Target

PDK

Receptor

CDK2/CyclinE; Chk1; c-Kit; PDK1

Chemical Name

1-Pyrrolidinecarboxamide, N-[3-[[5-iodo-4-[[3-[(2-thienylcarbonyl)amino]propyl]amino]-2-pyrimidinyl]amino]phenyl]

SMILES

O=C(N1CCCC1)NC2=CC=CC(NC3=NC=C(I)C(NCCCNC(C4=CC=CS4)=O)=N3)=C2

Molecular Formula

C23H26IN7O2S

CAS Number

702675-74-9

Product Categories/Family for BX795 biochemical

PI3K/Akt/mTOR signaling; Cancer

Product References and Citations for BX795 biochemical

1. Clark K, et al. J Biol Chem. 2009 May 22; 284 (21):14136-46.
2. Feldman RI, et al. J Biol Chem. 2005 May 20; 280 (20):19867-74.
3. Friemond ML, et al. Arthritis Rheumatol. 2017 Apr 20. doi: 10.1002/art.40122.

Other Notes

Small volumes of BX795 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for BX795 purchase

MBS3605694 is a biochemical targeting BX795.

BX795

Product Overview

Product Categories/Family for BX795 biochemical

Structure of BX795 biochemical

Related Product Information for BX795 biochemical

Product References and Citations for BX795 biochemical

Other Notes

Searchable Terms for BX795 purchase