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OSI-930

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3605783

A potent, orally active, dual inhibitor of c-Kit and VEGFR-2 (KDR) with IC50 of 15 nM and 9 nM, respectively. More details

$260 / 5 mg +1 FREE 8GB USB
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
OSI-930, Biochemical
Full Product Name
OSI-930
Product Synonym Names
OSI 930; OSI930
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20°C
Stability: >=2 years
Molecular Weight
443.44
Suitability
10mM in DMSO
Target
c-Kit
Receptor
C-Raf; CSF-1R; FLT1; Lck; VEGFR2 (KDR)
Chemical Name
2-Thiophenecarboxamide, 3-[(4-quinolinylmethyl)amino]-N-[4-(trifluoromethoxy)phenyl]
SMILES
O=C(C1=C(NCC2=CC=NC3=CC=CC=C23)C=CS1)NC4=CC=C(OC(F)(F)F)C=C4
Molecular Formula
C22H16F3N3O2S
CAS Number
728033-96-3
Pathway
Angiogenesis

Product Categories/Family for OSI-930 biochemical

Solid Tumors; Angiogenesis; Cancer

Structure of OSI-930 biochemical

OSI-930 Biochemical – Cat# MBS3605783

Product References and Citations for OSI-930 biochemical

1. Garton AJ, et al. Cancer Res. 2006 Jan 15; 66 (2):1015-24.
2. Yap TA, et al. Clin Cancer Res. 2013 Feb 15; 19 (4):909-19.
3. Patel JP, et al. Bioorg Med Chem Lett. 2011 Nov 1; 21 (21):6495-9.
4. Macpherson IR, et al. Eur J Cancer. 2013 Mar; 49 (4):782-9.

Other Notes

Small volumes of OSI-930 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for OSI-930 purchase

MBS3605783 is a biochemical targeting OSI-930.
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