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BMS-681

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3606153

A potent and orally bioavailable dual antagonist of CCR2 and CCR5 with binding IC50 of 0.7 nM and 2.4 nM, respectively. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
BMS-681, Biochemical
Full Product Name
BMS-681
Product Synonym Names
BMS 681; BMS681
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
491.603
Target
Chemokine Receptor
Receptor
Chemokine Receptor
Chemical Name
1-((1S, 2R, 4R)-4-(isopropyl(methyl)amino)-2-propylcyclohexyl)-3-((6-(trifluoromethyl)quinazolin-4-yl)amino)pyrrolidin-2-one
SMILES
CCCC1CC(CCC1N2CCC(C2=O)NC3=NC=NC4=C3C=C(C=C4)C(F)(F)F)N(C)C(C)C
Molecular Formula
C26H36F3N5O
CAS Number
847998-92-9
Dry Ice Shipment
Extra charge fee may add to your shipping cost as dry ice is required to ship this product.

Product Categories/Family for BMS-681 biochemical

GPCR/G Protein

Structure of BMS-681 biochemical

BMS-681 Biochemical – Cat# MBS3606153

Product References and Citations for BMS-681 biochemical

1. Zheng Y, et al. Nature. 2016 Dec 15; 540 (7633):458-461.
2. Carter PH, et al. ACS Med Chem Lett. 2015 Mar 4; 6 (4):439-44.

Other Notes

Small volumes of BMS-681 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for BMS-681 purchase

MBS3606153 is a biochemical targeting BMS-681.
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