Cebranopadol (GRT-6005)

Name: Cebranopadol (GRT-6005); MyBioSource
Brand: MyBioSource
SKU: MBS3606249
Price: 215 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3606249

Cebranopadol (GRT-6005, GRT6005) is a potent analgesic nociceptin/orphanin FQ peptide (NOP) and opioid receptor agonist with Ki/EC50 of 0.9/13 nM (human NOP receptor), 0.7/1.2 nM (mu-opioid receptor). More details

$215 / 2 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Cebranopadol, Biochemical

Full Product Name

Cebranopadol

Product Synonym Names

GRT-6005; GRT 6005; GRT6005

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

378.491

Suitability

DMSO: 6mg/mL
Water: Insoluble (<1mg/mL refers to the product slightly soluble or insoluble)

Target

Opioid Receptor

Receptor

NOP; u-opioidreceptor; kappa-opioidreceptor; delta-opioidreceptor

Chemical Name

(1r, 4r)-6'-fluoro-N, N-dimethyl-4-phenyl-4', 9'-dihydro-3'H-spiro[cyclohexane-1, 1'-pyrano[3, 4-b]indol]-4-amine

SMILES

CN(C)C1(CCC2(CC1)C3=C(CCO2)C4=C(N3)C=CC(=C4)F)C5=CC=CC=C5

Molecular Formula

C24H27FN2O

CAS Number

863513-91-1

Product Categories/Family for Cebranopadol biochemical

Pain; Endocrinology/Hormones; Neurological Disease

Product References and Citations for Cebranopadol biochemical

1. Linz K, et al. J Pharmacol Exp Ther. 2014 Jun; 349 (3):535-48.
2. Schunk S, et al. ACS Med Chem Lett. 2014 Jun 24; 5 (8):857-62.

Other Notes

Small volumes of Cebranopadol biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Cebranopadol purchase

MBS3606249 is a biochemical targeting Cebranopadol.