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GSK598809

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3606252

GSK598809 (GSK-598809) is a potent, selective, CNS penetrant and orally bioavailable dopamine D3 receptor antagonist with pKi of 8.9; displays >100-fold selectivity over D2 and H1 receptors. More details

$425 / 5 mg +1 FREE 8GB USB
Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
GSK598809, Biochemical
Full Product Name
GSK598809
Product Synonym Names
GSK 598809; GSK-598809
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
481.514
Suitability
DMSO: 83.33mg/mL (173.06mM)
Target
Dopamine Receptor
Receptor
Dopamine Receptor
Chemical Name
1-[2-Fluoro-4-(trifluoromethyl)phenyl]-3-[3-[[4-methyl-5-(4-methyl-1, 3-oxazol-5-yl)-4H-1, 2, 4-triazol-3-yl]thio]propyl]-3-azabicyclo[3.1.0]hexane
SMILES
CC1=C(OC=N1)C2=NN=C(N2C)SCCCN3CC4CC4(C3)C5=C(C=C(C=C5)C(F)(F)F)F
Molecular Formula
C22H23F4N5OS
CAS Number
863680-45-9

Product Categories/Family for GSK598809 biochemical

Other Disease; GPCR/G Protein; Other Indications

Structure of GSK598809 biochemical

GSK598809 Biochemical – Cat# MBS3606252

Product References and Citations for GSK598809 biochemical

1. Micheli F, et al. J Med Chem. 2010 Jan 14; 53 (1):374-91.
2. AppelnM, et al. J Pharmacol Exp Ther. 2015 Sep; 354 (3):484-92.
3. Dodds CM, et al. Appetite. 2012 Aug; 59 (1):27-33.
4. Searle G, et al. Biol Psychiatry. 2010 Aug 15; 68 (4):392-9.

Other Notes

Small volumes of GSK598809 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GSK598809 purchase

MBS3606252 is a biochemical targeting GSK598809.
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