Linsitinib (ASP-7487)

Name: Linsitinib (ASP-7487); MyBioSource
Brand: MyBioSource
SKU: MBS3606298
Price: 215 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3606298

Linsitinib (ASP-7487, OSI-906) is a potent, selective, orally active, dual IGF-1R/insulin receptor inhibitor with IC50 of 35/75 nM, respectively. More details

$215 / 2 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Linsitinib, Biochemical

Full Product Name

Linsitinib

Product Synonym Names

ASP-7487; ASP 7487; OSI-906; OSI906

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

421.4937

Suitability

10mM in DMSO

Target

IGF-1R

Receptor

IGF-1R; InsulinReceptor; IRR

Chemical Name

Cyclobutanol, 3-[8-amino-1-(2-phenyl-7-quinolinyl)imidazo[1, 5-a]pyrazin-3-yl]-1-methyl-, cis

SMILES

O[C@@]1(C)C[C@H](C2=NC(C3=CC=C4C=CC(C5=CC=CC=C5)=NC4=C3)=C6C(N)=NC=CN62)C1

Molecular Formula

C26H23N5O

CAS Number

867160-71-2

Product Categories/Family for Linsitinib biochemical

Liver Cancer; Angiogenesis; Cancer

Product References and Citations for Linsitinib biochemical

1. Mulvihill MJ, et al. Future Med Chem. 2009 Sep; 1 (6):1153-71.
2. Pitts TM, et al. Clin Cancer Res. 2010 Jun 15; 16 (12):3193-204.
3. Buck E, et al. Mol Cancer Ther. 2010 Oct; 9 (10):2652-64.
4. Kuhn DJ, et al. Blood. 2012 Oct 18; 120 (16):3260-70.

Other Notes

Small volumes of Linsitinib biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Linsitinib purchase

MBS3606298 is a biochemical targeting Linsitinib.