• Call +1.858.633.0165 or Fax +1.858.633.0166 or Contact Us

BL5923

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3606599

BL5923 (BL-5923) is a potent, highly specific, orally available inhibitor of CCR1 with IC50 of 20.4 and 22.8 nM for human and mouse CCR1, resepctively. More details

Please Inquire
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
BL5923, Biochemical
Full Product Name
BL5923
Product Synonym Names
BL 5923; BL-5923
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
487.956
Target
Chemokine Receptor
Receptor
Chemokine Receptor
Chemical Name
(E)-N-(5-chloro-2-(3-(9-(4-fluorobenzyl)-3-oxa-7, 9-diazabicyclo[3.3.1]nonan-7-yl)-3-oxoprop-1-en-1-yl)-4-methoxyphenyl)acetamide
SMILES
CC(=O)NC1=CC(=C(C=C1C=CC(=O)N2CC3COCC(C2)N3CC4=CC=C(C=C4)F)OC)Cl
Molecular Formula
C25H27ClFN3O4
CAS Number
921208-19-7

Product Categories/Family for BL5923 biochemical

GPCR/G Protein

Structure of BL5923 biochemical

BL5923 Biochemical – Cat# MBS3606599

Product References and Citations for BL5923 biochemical

1. Kitamura T, et al. Proc Natl Acad Sci U S A. 2010 Jul 20; 107 (29):13063-8.
2. Revesz L, et al. Bridged piperazines and piperidines as CCR1 antagonists with oral activity in models of arthritis and multiple sclerosis. Lett Drug Des Discov. 2006; 3:689-694.
3. Bignon A, et al. J Immunol. 2014 Feb 1; 192 (3):886-96.
4. Lionakis MS, et al. Antimicrob Agents Chemother. 2017 Feb 23; 61 (3). pii: e02365-16.

Other Notes

Small volumes of BL5923 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for BL5923 purchase

MBS3606599 is a biochemical targeting BL5923.
Request a Quote

Please fill out the form below and our representative will get back to you shortly.

MBS000000
Contact Us

Please fill out the form below and our representative will get back to you shortly.

MBS000000