GSK-461364A Biochemical – Cat# MBS3606648

GSK-461364 (GSK-461364A)

Name: GSK-461364A; MyBioSource
Brand: MyBioSource
SKU: MBS3606648
Price: 235 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3606648

A potent, selective, and reversible ATP-competitive PLK1 inhibitor with Ki of 2.2 nM. More details

$235 / 2 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

GSK-461364, Biochemical

Full Product Name

GSK-461364

Product Synonym Names

GSK-461364A

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

543.6038

Suitability

10mM in DMSO

Target

PLK

Receptor

PLK1

Chemical Name

2-Thiophenecarboxamide, 5-[6-[(4-methyl-1-piperazinyl)methyl]-1H-benzimidazol-1-yl]-3-[(1R)-1-[2-(trifluoromethyl)phenyl]ethoxy]

SMILES

O=C(C1=C(O[C@@H](C2=CC=CC=C2C(F)(F)F)C)C=C(N3C=NC4=CC=C(CN5CCN(C)CC5)C=C34)S1)N

Molecular Formula

C27H28F3N5O2S

CAS Number

929095-18-1

Product Categories/Family for GSK-461364 biochemical

Blood cancer; Cell Cycle/DNA Damage; Cancer

Product References and Citations for GSK-461364 biochemical

1. Olmos D, et al. Clin Cancer Res. 2011 May 15; 17 (10):3420-30.
2. Gilmartin AG, et al. Cancer Res. 2009 Sep 1; 69 (17):6969-77.
3. Degenhardt Y, et al. Mol Cancer Ther. 2010 Jul; 9 (7):2079-89.

Other Notes

Small volumes of GSK-461364 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GSK-461364 purchase

MBS3606648 is a biochemical targeting GSK-461364.